83846-83-7 Ketanserin (+)-tartrate salt AKSci V1493
 
 
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  V1493    
Ketanserin (+)-tartrate salt, >98% (HPLC)
 
3-(2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl)-2,4(1H,3H)-quinazolinedione (+)-tartrate salt, R 41468 (+)-tartrate salt
IDENTITY
CAS Number:83846-83-7
MDL Number:MFCD11864992
MF:C26H28FN3O9
MW:545.51
EINECS:281-062-8
SPECIFICATIONS & PROPERTIES
Min. Purity Spec:>98% (HPLC)
Physical Form (at 20°C):Solid
Melting Point:163-168°C
Long-Term Storage:Store long-term at 2-8°C
DOT/IATA TRANSPORT INFORMATION
UN #:UN2811
Hazard Class:6.1; Poison
Packing Group:III
A hazmat fee may apply to certain package sizes. Please check pricing table for an indicator of applicable hazmat fees.

BIOLOGICAL INFO
Application(s):A selective serotonin agonist

REVIEW
 Ketanserin tartrate is a salt of Ketanserin. Ketanserin is reported to have a high affinity for multiple G protein-coupled receptors, such as serotonin receptors. Ketanserin is a selective SR-2/SR-1C antagonist. It has been used to distinguish between SR-1D and SR-1B subtypes. Additional studies have noted that Ketanserin is able to differentiate between recombinant human forms of these receptors with a higher affinity for SR-1Dalfa receptors compared to SR-1Dbeta receptors. Ketanserin tartrate is an inhibitor of SR-2A and SR-2C.

REFERENCES
[1]Van Nueten, J.M., et al. 1981. J. Pharmacol. Exp. Ther. 218: 217-230. PMID: 6113280
[2] Leysen, J.E., et al. 1982. Mol. Pharmacol. 21: 301-314. PMID: 7099138

GLOBALLY HARMONIZED SYSTEM (GHS)

Pictograms

Signal Word
Danger

Hazard Statements
H301

Precautionary Statements
P264; P270; P301+P310; P321; P330; P405; P501

RELATED PRODUCTS
K261Ketanserin
V1493Ketanserin (+)-tartrate salt

Current as of April 25, 2024


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CATEGORIES
 APIs and Bioactives > Hypertension


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